HEPPERLE M ET AL: "Mono N-arylation of piperazine(III): metal-catalyzed N-arylation and its application to the novel preparations of the antifungal posaconazole and its advanced intermediate", TETRAHEDRON LETTERS, PERGAMON, GB, vol. 43, no. 18, 29 April 2002 (2002-04-29), pages 3359-3363, XP004349385, ISSN: 0040-4039, DOI: 10.1016/S0040-4039(02)00556-7 (B1)

SAKSENA A K ET AL: "Stereoselective Grignard additions to N-formyl hydrazone: a concise synthesis of Noxafil<R> side chain and a synthesis of Noxafil<R>", TETRAHEDRON LETTERS, PERGAMON, GB, vol. 45, no. 44, 25 October 2004 (2004-10-25), pages 8249-8251, XP004591093, ISSN: 0040-4039, DOI: 10.1016/J.TETLET.2004.09.028 (B1)

PAUL BOWYER ET AL: "Environmental fungicides and triazole resistance in Aspergillus", PEST MANAGEMENT SCIENCE, vol. 70, no. 2, 5 February 2014 (2014-02-05), pages 173-178, XP055169575, ISSN: 1526-498X, DOI: 10.1002/ps.3567 cited in the application (B1)