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Org.nummer: 982702887
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2011.06.10, US 201161495773 P
KATTAR S D ET AL: "Parallel medicinal chemistry approaches to selective HDAC1/HDAC2 inhibitor (SHI-1:2) optimization", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, ELSEVIER SCIENCE, GB, vol. 19, no. 4, 15 February 2009 (2009-02-15), pages 1168-1172, XP025937239, ISSN: 0960-894X, DOI: 10.1016/J.BMCL.2008.12.083 [retrieved on 2009-02-10] (B1)
JP-A- 8 283 246 (B1)
O'BRIEN D E ET AL: "Pyrimidines. XI. Structural Variations of 2,4-Diamino-6-(halogenoanilino)-5.nitrosop yrimidines", JOURNAL OF MEDICINAL CHEMISTRY,, vol. 6, no. 5, 11 September 1963 (1963-09-11), pages 467-471, XP002647746, (B1)
PEGIADOU: "The synthesis and characterization of new polymerizable pyrimidines: Immobilization of the monomers onto hydrophilic graft copolymeric supports through radiation-induced copolymerization-grafting", JOURNAL OF APPLIED POLYMER SCIENCE, vol. 70, no. 2, 1 January 1998 (1998-01-01), page 211, XP55048115, ISSN: 0021-8995 (B1)
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TRAVERSO J J ET AL: "THE SYNTHESIS AND PHARMACOLOGICAL ACTIVITIES OF AMIDE, SULFAMIDE, AND UREA DERIVATIVES OF 4,6-DIAMINOPYRIMIDINES", JOURNAL OF MEDICINAL AND PHARMACEUTICAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY. EASTON, US, vol. 5, 1 July 1962 (1962-07-01), pages 808-815, XP000653960, DOI: 10.1021/JM01239A015 (B1)
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VISHWAKARMA J N ET AL: "Reactions of Polarized Keten S,N-Acetals with Guanidine: A Facile General Route to Novel 5,6-Substituted 2-Amino-4-N-alkyl/aryl/N-azacycloalkylamin opyrimidines", INDIAN JOURNAL OF CHEMISTRY. SECTION B: ORGANIC AND MEDICINAL CHEMISTRY, COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (C S I R), IN, vol. 24, 1 January 1985 (1985-01-01), pages 466-471, XP009162452, ISSN: 0376-4699 (B1)
WEN SONG YUE ET AL: "A Concise Synthesis of All Four Possible Benzo[4,5]furopyridines via Palladium-Mediated Reactions", ORGANIC LETTERS, vol. 4, no. 13, 1 June 2002 (2002-06-01), pages 2201-2203, XP55042429, ISSN: 1523-7060, DOI: 10.1021/ol0260425 (B1)
WHITEHEAD C W & TRAVERSO J J: "Diuretics. III. 4,6-Diaminopyrimidines", JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, ACS PUBLICATIONS, US, vol. 80, 5 May 1958 (1958-05-05), pages 2185-2189, XP002081959, ISSN: 0002-7863, DOI: 10.1021/JA01542A038 (B1)
WILLIAM W. PAUDLER ET AL: "Bromination of some pyridine and diazine N-oxides", THE JOURNAL OF ORGANIC CHEMISTRY, vol. 48, no. 7, 1 April 1983 (1983-04-01), pages 1064-1069, XP55047990, ISSN: 0022-3263, DOI: 10.1021/jo00155a027 (B1)
WO-A1-2007/089512 (B1)
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WO-A1-2009/158571 (B1)
WO-A1-2010/057126 (B1)
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WO-A1-2011/029043 (B1)
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ZHANG Y M ET AL: "Synthesis of pyrimido[4,5-b]indoles and benzo[4,5]furo[2,3-d]pyrimidines via palladium-catalyzed intramolecular arylation", TETRAHEDRON LETTERS, ELSEVIER, AMSTERDAM, NL, vol. 43, no. 46, 11 November 2002 (2002-11-11), pages 8235-8239, XP027330566, ISSN: 0040-4039 [retrieved on 2002-11-11] (B1)
ACKERMANN H ET AL: "Konstitution und Reaktionsfaehigkeit von Trichlor-pyrimidylamino-Verbindungen", HELVETICA CHIMICA ACTA, VERLAG HELVETICA CHIMICA ACTA, BASEL, CH, vol. 45, no. 5, 1 January 1962 (1962-01-01), pages 1683-1698, XP009162477, ISSN: 0018-019X (B1)
ALAN C. SPIVEY ET AL: "Atropisomeric [alpha]-methyl substituted analogues of 4-(dimethylamino)pyridine: synthesis and evaluation as acyl transfer catalysts", JOURNAL OF THE CHEMICAL SOCIETY, PERKIN TRANSACTIONS 1, no. 15, 1 January 2001 (2001-01-01), pages 1785-1794, XP55048017, ISSN: 1472-7781, DOI: 10.1039/b103385a (B1)
ALLA BESSMERTNYKH ET AL: "Efficient Palladium-Catalyzed Synthesis of Aminopyridyl Phosphonates from Bromopyridines and Diethyl Phosphite", SYNTHESIS, vol. 2008, no. 10, 1 May 2008 (2008-05-01) , pages 1575-1579, XP55048046, ISSN: 0039-7881, DOI: 10.1055/s-2008-1072570 (B1)
ARTHUR P. PHILLIPS ET AL: "Syntheses of 1,3-Diazaphenothiazines.1 I.", THE JOURNAL OF ORGANIC CHEMISTRY, vol. 28, no. 6, 1 June 1963 (1963-06-01), pages 1488-1490, XP55042306, ISSN: 0022-3263, DOI: 10.1021/jo01041a012 (B1)
ATWAL K S ET AL: "Synthesis and biological activity of 5-aryl-4-(4-(5-methyl-1H-imidazol-4-yl)pip eridin-1-yl)pyrimidine analogs as potent, highly selective, and orally bioavailable NHE-1 inhibitors", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, ELSEVIER SCIENCE, GB, vol. 16, no. 18, 15 September 2006 (2006-09-15), pages 4796-4799, XP027966643, ISSN: 0960-894X [retrieved on 2006-09-15] (B1)
BIRESSI ET AL: "Su Alcune 5-Fluoro-6-Anilino-Amminopirimidine", BOLLETTINO CHIMICO FARMACEUTICO, SOCIETA EDITORIALE FARMACEUTICA, MILANO, IT, vol. 105, 1 January 1966 (1966-01-01), pages 660-665, XP009162478, ISSN: 0006-6648 (B1)
BONGKOCH TARNCHOMPOO ET AL: "Development of 2,4-Diaminopyrimidines as Antimalarials Based on Inhibition of the S108N and C59R+S108N Mutants of Dihydrofolate Reductase from Pyrimethamine-Resistant Plasmodium f alciparum", JOURNAL OF MEDICINAL CHEMISTRY, vol. 45, no. 6, 1 March 2002 (2002-03-01), pages 1244-1252, XP55048052, ISSN: 0022-2623, DOI: 10.1021/jm010131q (B1)
B]TTELMANN B ET AL: "4-(3,4-DIHYDRO-1H-ISOQUINOLIN-2YL)-PYRIDI NES AND 4-(3,4-DIHYDRO-1H-ISOQUINOLIN-2-YL)-QUINOL INES AS POTENT NR1/2B SUBTYPE SELECTIVE NMDA RECEPTOR ANTAGONISTS", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, ELSEVIER SCIENCE, GB, vol. 13, 1 January 2003 (2003-01-01), pages 1759-1762, XP003009973, ISSN: 0960-894X, DOI: 10.1016/S0960-894X(03)00232-4 (B1)
C. BARILLARI ET AL: "Solid Phase Synthesis of Diamino-Substituted Pyrimidines", EUR. J. ORG. CHEM., 1 January 2001 (2001-01-01), pages 4737-4741, XP55044047, (B1)
CHANG SUNG HONG ET AL: "Synthesis of Aromatic Ring Fused Pyrrole Derivatives by Palladium-catalyzed Annulation of o-Iodoarylamines with Allyl Acetate", HETEROCYCLES, ELSEVIER SCIENCE PUBLISHERS B.V. AMSTERDAM, NL, vol. 63, no. 3, 1 January 2004 (2004-01-01), pages 631-639, XP001526304, ISSN: 0385-5414 (B1)
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EP-A1- 0 471 297 (B1)
EP-A1- 1 348 706 (B1)
HURST D T: "Application of the Elbs Persulfate Oxidation to the Preparation of 5-Hydroxypyrimidines", AUSTRALIAN JOURNAL OF CHEMISTRY, CSIRO, AU, vol. 36, 1 January 1983 (1983-01-01), pages 1285-1289, XP009088310, ISSN: 0004-9425 (B1)
IWAKI ET AL: "Novel synthetic strategy of carbolines via palladium-catalized amination and arylation reaction", JOURNAL OF THE CHEMICAL SOCIETY, PERKIN TRANSACTIONS 1, CHEMICAL SOCIETY, LETCHWORTH; GB, 1 January 1999 (1999-01-01), pages 1505-1510, XP002458090, ISSN: 0300-922X, DOI: 10.1039/A901088B (B1)
JANG M Y ET AL: "Synthesis of novel 5-amino-thiazolo[4,5-d]pyrimidines as E. coli and S. aureus SecA inhibitors", BIOORGANIC & MEDICINAL CHEMISTRY, PERGAMON, GB, vol. 19, no. 1, 1 January 2011 (2011-01-01), pages 702-714, XP027577807, ISSN: 0968-0896 [retrieved on 2010-12-28] (B1)
JONATHAN LARGE ET AL: "Synthesis of Trisubstituted Pyrimidines by Regioselective S N Ar and Suzuki Reactions of Polyhalopyrimidines", SYNLETT, vol. 2006, no. 6, 1 April 2006 (2006-04-01), pages 861-864, XP55048077, ISSN: 0936-5214, DOI: 10.1055/s-2006-939050 (B1)
KOSARY J ET AL: "preparation of pyrimidine derivatives with potential cardiotonic activity", ACTA PHARMACEUTICA HUNGARICA, HUNGARICAN PHARMACEUTICAL ASSOCIATION, BUDAPEST, HU, vol. 59, 1 January 1989 (1989-01-01), pages 241-247, XP002119936, ISSN: 0001-6659 (B1)
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Til betaling:
En ordre på saken er opprettet av: ANAQUA ANAQUA (20.05.2025 09:56:08): Opprettet, ikke betalt
Betalingshistorikk:
Beskrivelse / Fakturanummer | Betalingsdato | Beløp | Betaler | Status |
---|---|---|---|---|
Årsavgift 13. avg. år (EP) | 2024.06.11 | 5460 | CPA GLOBAL LIMITED | Betalt og godkjent |
Årsavgift 12. avg. år (EP) | 2023.06.08 | 3850 | CPA GLOBAL LIMITED | Betalt og godkjent |
Årsavgift 11. avg. år (EP) | 2022.06.09 | 3500 | CPA GLOBAL LIMITED | Betalt og godkjent |
32206887 expand_more expand_less | 2022.05.18 | 5500 | ZACCO NORWAY AS | Betalt |
Valideringsgebyr EP-patent
5500 = 1 X 5500
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