DATABASE EMBASE [Online] ELSEVIER SCIENCE PUBLISHERS, AMSTERDAM, NL; 1998, BONSMANN U ET AL: "Metabolisation and receptor affinity of topically applied esters of glucocorticoids", XP002788474, Database accession no. EMB-1998329776 & BONSMANN U ET AL: "Metabolisation and receptor affinity of topically applied esters of glucocorticoids", H+G ZEITSCHRIFT FUR HAUTKRANKHEITEN 1998 DE, vol. 73, no. 9, 1998, pages 581-590, ISSN: 0301-0481 (B1)

DATABASE HCAPLUS, [Online] 1 January 1979 (1979-01-01), CUTLER GORDON B ET AL: "11-Deoxycortisol: a glucocorticoid antagonist in vivo", XP002749428, retrieved from HCAPLUS; STN Database accession no. 1979-469056 & CUTLER G B JR ET AL: "11-Deoxycortisol: a glucocorticoid antagonist in vivo.", ENDOCRINOLOGY JUN 1979, vol. 104, no. 6, June 1979 (1979-06), pages 1839-1844, ISSN: 0013-7227 (B1)

FERRABOSCHI P ET AL: "Lipase-catalyzed preparation of corticosteroid 17@a-esters endowed with antiandrogenic activity", TETRAHEDRON LETTERS, ELSEVIER, AMSTERDAM, NL, vol. 49, no. 31, 28 July 2008 (2008-07-28) , pages 4610-4612, XP022757401, ISSN: 0040-4039, DOI: 10.1016/J.TETLET.2008.05.086 [retrieved on 2008-05-23] (B1)

WO-A2-2009/019138 (B1)

PATRIZIA FERRABOSCHI ET AL: "A full conformational characterization of antiandrogen cortexolone-17[alpha]-propionate and related compounds through theoretical calculations and nuclear magnetic resonance spectroscopy", MEDCHEMCOMM, vol. 5, no. 7, 1 January 2014 (2014-01-01) , pages 904-914, XP55224342, United Kingdom ISSN: 2040-2503, DOI: 10.1039/C4MD00049H (B1)

SEAN EKINS ET AL: "Challenges Predicting Ligand-Receptor Interactions of Promiscuous Proteins: The Nuclear Receptor PXR", PLOS COMPUTATIONAL BIOLOGY, vol. 5, no. 12, 11 December 2009 (2009-12-11), pages e1000594-1, XP055549623, DOI: 10.1371/journal.pcbi.1000594 -& Sean Ekins ET AL: "Challenges Predicting Ligand-Receptor Interactions of Promiscuous Proteins: The Nuclear Receptor PXR", PLoS Computational Biology, 11 December 2009 (2009-12-11), page e1000594, XP055549646, DOI: 10.1371/journal.pcbi.1000594 Retrieved from the Internet: URL:https://journals.plos.org/ploscompbiol /article/file?id=10.1371/journal.pcbi.1000 594.s002&type=supplementary [retrieved on 2019-01-30] -& Sean Ekins ET AL: "Challenges Predicting Ligand-Receptor Interactions of Promiscuous Proteins: The Nuclear Receptor PXR", PLoS Computational Biology, 11 December 2009 (2009-12-11), page e1000594, XP055549647, DOI: 10.137 (B1)

US-A- 3 152 154 (B1)

GIUSEPPE CELASCOA ET AL: "Pharmacological Profile of 9,11-Dehydrocortexolone 17[alpha]-Butyrate (CB-03-04), a New Androgen Antagonist with Antigonadotropic Activity", ARZNEIMITTEL FORSCHUNG. DRUG RESEARCH, ECV EDITIO CANTOR VERLAG, AULENDORF, DE, vol. 55, no. 10, 1 January 2005 (2005-01-01), pages 581-587, XP008175216, ISSN: 0004-4172, DOI: 10.1055/S-0031-1296908 (B1)